A novel anabolic agent: A simvastatin analogue without HMG-CoA reductase inhibitory activity

Kuang Chan Hsieh, Chai Lin Kao, Chien Wei Feng, Zhi Hong Wen, Hsin Fang Chang, Shu Chun Chuang, Gwo Jaw Wang, Mei Ling Ho, Shou Mei Wu*, Je Ken Chang, Hui Ting Chen

*此作品的通信作者

研究成果: Article同行評審

4 引文 斯高帕斯(Scopus)

摘要

For the first time, structural information regarding the role of simvastatin in bone anabolism is described, and a bone-specific statin is introduced. Polyaspartate-conjugated simvastatin was synthesized by solid-phase synthesis with the assistance of microwave irradiation. It displays significant bone targeting and bone formation with less toxicity than simvastatin.

原文English
頁(從 - 到)4376-4379
頁數4
期刊Organic Letters
16
發行號17
DOIs
出版狀態Published - 5 9月 2014

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